A tritiated tetrazine based on a phenyl/pyridyl core structure was successfully radiolabeled with NaBT₄ by reducing an aldehyde moiety. The synthon was effectively employed to label an antibody in vitro with pretargeted autoradiography.

中文翻译：

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第一种氚化四嗪的开发：促进蛋白质的氚化

基于苯基/吡啶基核心结构的氚化四嗪通过还原醛部分成功地用 NaBT _{4进行了放射性标记。}该合成子被有效地用于通过预靶向放射自显影在体外标记抗体。